Fig. 1 · Structure
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LY2940094 tartrate
NOP Receptor Antagonist
LY2940094 tartrate is a potent and selective antagonist of the nociceptin/orphanin FQ (NOP) receptor, characterized by a high binding affinity (Ki=0.105 nM) and effective antagonistic potency (Kb=0.166 nM). This compound exhibits significant brain penetration and is orally bioavailable, making it suitable for in vivo studies. LY2940094 tartrate has demonstrated efficacy in reducing ethanol self-administration and seeking behaviors in animal models, providing valuable insights for research in addiction and neuropharmacology.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Antagonist |
| CAS Number | 1307245-87-9 |
| Applications | NOP Receptor Antagonist |
| Formula | C26H29ClF2N4O8S |
| Molecular Weight | 631.05 |
| Synonyms | BTRX-246040 tartrate |
| SMILES | OCC1=CC=CN=C1N2N=C(C)C(CN3CCC4(C5=C(C=C(Cl)S5)C(F)(F)CO4)CC3)=C2.O=C(O)[C@H](O)[C@@H](O)C(O)=O |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.