Fig. 1 · Structure
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M77976
PDK4 Inhibitor
M77976 is a selective ATP-competitive inhibitor of pyruvate dehydrogenase kinase isoform 4 (PDK4), exhibiting an IC50 of 648 μM. This compound plays a critical role in metabolic research, particularly in the study of obesity and diabetes, by modulating glucose metabolism and energy homeostasis. M77976 is valuable for exploring the therapeutic potential of targeting PDK4 in metabolic disorders.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Inhibitor |
| CAS Number | 394237-61-7 |
| Applications | PDK4 Inhibitor |
| Formula | C17H16N2O3 |
| Molecular Weight | 296.32 |
| SMILES | COC1=CC=C(C=C1)C2=C(NN=C2C3=CC=C(C=C3O)O)C |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.