Fig. 1 · Structure
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Metoprine
HMT Inhibitor
Metoprine is a potent inhibitor of histamine N-methyltransferase (HMT), effectively increasing brain histamine levels by blocking its enzymatic activity. As a diaminopyrimidine derivative, Metoprine is capable of crossing the blood-brain barrier, making it suitable for neurological research. Additionally, it exhibits antifolate and antitumor properties, positioning it as a valuable tool for studying tumor biology and histamine-related functions in various biological systems.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Inhibitor |
| CAS Number | 7761-45-7 |
| Applications | HMT Inhibitor |
| Formula | C11H10Cl2N4 |
| Molecular Weight | 269.13 |
| Synonyms | BW 197U |
| SMILES | CC1=C(C(N)=NC(N)=N1)C2=CC=C(C(Cl)=C2)Cl |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.