Fig. 1 · Structure
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mGlu4 receptor agonist 1
mGlu4 Receptor Agonist
mGlu4 receptor agonist 1 is a potent positive allosteric modulator targeting the mGlu4 receptor, exhibiting an EC50 value of 308 nM. This compound has demonstrated significant anxiolytic and antipsychotic-like activity, making it a valuable tool for research into neuropharmacology and the modulation of glutamatergic processes. Its unique mechanism of action offers potential insights into the treatment of anxiety and psychotic disorders.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Modulator |
| CAS Number | 1678501-16-0 |
| Applications | mGlu4 Receptor Agonist |
| Formula | C21H15ClN4O2 |
| Molecular Weight | 390.82 |
| SMILES | CC1=CC(NC(C2=CC=CC=N2)=O)=CC=C1C3=NOC(C4=C(C=CC=C4)Cl)=N3 |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.