MK-3207

Catalog No.: A15165

CGRP Receptor antagonist

MK-3207

MK-3207 Chemical Structure

CAS NO. 957118-49-9

MK-3207 is a potent and orally bioavailable CGRP receptor antagonist (IC50= 0.12 nM; Ki value= 0.024 nM); highly selective versus human AM1, AM2, CTR, and AMY3.

Availability: In stock

Package Price Qty
10 mg
$200.00
25 mg
$380.00
50 mg
$650.00
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Biological Activity

MK-3207 is a potent and orally bioavailable CGRP receptor antagonist (IC50= 0.12 nM; Ki value= 0.024 nM); highly selective versus human AM1, AM2, CTR, and AMY3.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 17.93 mL 89.67 mL 179.34 mL
0.5 mM 3.59 mL 17.93 mL 35.87 mL
1 mM 1.79 mL 8.97 mL 17.93 mL
5 mM 0.36 mL 1.79 mL 3.59 mL

*The above data is based on the productmolecular weight 557.59. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A15165
Actions Antagonist
CAS No. 957118-49-9
Formula C31H29F2N5O3
M. Wt 557.59
Purity >98%
Synonyms MK3207, MK 3207
SMILES C1CCC2(C1)C(=O)N(C(CN2)C3=CC(=CC(=C3)F)F)CC(=O)NC4=CC5=C(CC6(C5)C7=C(NC6=O)N=CC=C7)C=C4
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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