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MK2-IN-5

MAPK Inhibitor

MK2-IN-5 is a potent MAPK inhibitor that functions as a pseudosubstrate with a Ki value of 8 μM. By targeting the protein interaction domain within the MAPK pathway, MK2-IN-5 effectively inhibits the phosphorylation of HSP25 and HSP27. This compound is useful for research applications focused on cellular signaling and stress response mechanisms.

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Specifications

Manufacturer	Adooq Bioscience
Actions	Inhibitor
CAS Number	474713-20-7
Applications	MAPK Inhibitor
Formula	C₆₁H₁₁₃N₂₁O₁₆
Molecular Weight	1396.68
Synonyms	Hsp25 kinase inhibitor; Mk2 pseudosubstrate
SMILES	[C@H](C(N[C@H](C(N[C@H](C(NCC(N[C@H](C(N[C@H](C(N[C@H](C(O)=O)C)=O)C)=O)C(C)C)=O)=O)CC(C)C)=O)CCC(N)=O)=O)(NC([C@@H](NC([C@@H](NC([C@@H](NC([C@@H](NC([C@@H](NC([C@H](CCCCN)N)=O)CCCCN)=O)CCCCN)=O)C)=O)CC(C)C)=O)CC(N)=O)=O)CCCNC(=N)N

Storage & Solubility

In Vitro Solubility

Reported Solubility

No reported solubility data are available for this product.

Preparing Stock Solutions

Stock preparation is unavailable for this product molecular weight.

Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.

Storage

Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.