Fig. 1 · Structure
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ML00253764
MC4R Antagonist
ML00253764 is a selective antagonist of the melanocortin receptor 4 (MC4R). It induces apoptosis through the inhibition of ERK1/2 and Akt phosphorylation pathways, demonstrating notable anticancer activity. This compound is valuable for research focused on cancer biology and the modulation of melanocortin signaling pathways.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Antagonist |
| CAS Number | 681847-92-7 |
| Applications | MC4R Antagonist |
| Formula | C18H18BrFN2O |
| Molecular Weight | 377.25 |
| SMILES | FC1=C(CCC2=CC(Br)=CC=C2OC)C(C3=NCCN3)=CC=C1 |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.