MMSET-IN-1

Catalog No.: A18860

SET domain inhibitor

MMSET-IN-1

MMSET-IN-1 Chemical Structure

CAS NO. 1998139-29-9

MMSET-IN-1 is a multiple myeloma SET domain (MMSET, aka NSD2/WHSC1) inhibitor against SETD2 and MMSET with IC50s of 0.49 and 3.3 μM, respectively. MMSET-IN-1 has a Kd of 1.6 μM for MMSET.

Availability: In stock

Package Price Qty
1 mg
$320.00
5 mg
$960.00
10 mg
$1,600.00
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Biological Activity

MMSET-IN-1 is a multiple myeloma SET domain (MMSET, aka NSD2/WHSC1) inhibitor against SETD2 and MMSET with IC50s of 0.49 and 3.3 μM, respectively. MMSET-IN-1 has a Kd of 1.6 μM for MMSET.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 23.61 mL 118.07 mL 236.14 mL
0.5 mM 4.72 mL 23.61 mL 47.23 mL
1 mM 2.36 mL 11.81 mL 23.61 mL
5 mM 0.47 mL 2.36 mL 4.72 mL

*The above data is based on the productmolecular weight 423.47. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A18860
Actions Inhibitor
CAS No. 1998139-29-9
Formula C18H29N7O5
M. Wt 423.47
Purity >98%
SMILES O=C(O)[[email protected]@H](N)CCC(NCCC)C[[email protected]]1O[[email protected]@H](N2C=NC3=C(N)N=CN=C23)[[email protected]](O)[[email protected]@H]1O
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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