Mozavaptan

Catalog No.: A16622

nonpeptide vasopressin V2 receptor antagonist

Mozavaptan

Mozavaptan Chemical Structure

CAS NO. 137975-06-5

Mozavaptan (OPC31260) is a orally effective, nonpeptide vasopressin V2 receptor antagonist with an IC50 of 14 nM.

Availability: In stock

Package Price Qty
10 mg
$54.00
25 mg
$108.00
50 mg
$186.00
100 mg
$318.00
Custom Size Get quote

Free Overnight Delivery on orders over $500

Next day delivery by 10:00 a.m. Order now.

Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

Mozavaptan (OPC31260) is a orally effective, nonpeptide vasopressin V2 receptor antagonist with an IC50 of 14 nM.
In vitro (25°C) DMSO 1 mg/mL (2.33 mM)
Water Insoluble
Ethanol 1 mg/mL (2.33 mM)
In vivo 30% propylene glycol, 5% Tween 80, 65% D5W 28 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 23.39 mL 116.95 mL 233.9 mL
0.5 mM 4.68 mL 23.39 mL 46.78 mL
1 mM 2.34 mL 11.69 mL 23.39 mL
5 mM 0.47 mL 2.34 mL 4.68 mL

*The above data is based on the productmolecular weight 427.54. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A16622
Actions Antagonist
CAS No. 137975-06-5
Formula C27H29N3O2
M. Wt 427.54
Purity >98%
SMILES CC1=CC=CC=C1C(NC2=CC=C(C(N3C(C=CC=C4)=C4C(N(C)C)CCC3)=O)C=C2)=O
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

Product Tags

Product Tags

Use spaces to separate tags. Use single quotes (') for phrases.

Product Questions

Product Questions

No Questions
Keywords:buy Mozavaptan | Mozavaptan Supplier | purchase | cost | manufacturer | order | distributor | buy 137975-06-5| 137975-06-5 Supplier | purchase 137975-06-5 | 137975-06-5 cost | 137975-06-5 manufacturer | order 137975-06-5 | 137975-06-5 distributor
Rewards