Fig. 1 · Structure
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MPCI
MC4R Antagonist
MPCI is a selective antagonist of the melanocortin-4 receptor (MC4R), exhibiting pharmacological chaperone activity. With a Ki value of 0.218 μM determined in HEK293 cells expressing human MC4R, MPCI is valuable in researching the mechanisms underlying MC4R-deficient obesity. This compound can facilitate studies on metabolic regulation and potential therapeutic approaches for related disorders.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Antagonist |
| CAS Number | 884538-31-2 |
| Applications | MC4R Antagonist |
| Formula | C25H32BrFN4O2 |
| Molecular Weight | 519.45 |
| SMILES | O=C(C1=CC=CC(F)=C1CCC2=CC(Br)=CC=C2OC)NC(NCC3CCN(CC3)CC)=N |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.