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MrgprX2 antagonist-10

MrgprX2 Antagonist

MrgprX2 antagonist-10 is a potent antagonist of the Mas-related G protein-coupled receptor X2 (MrgprX2), exhibiting an IC50 of less than 100 nM. This compound is valuable for researching the role of MrgprX2 in various inflammatory diseases, providing insights into potential therapeutic strategies targeting this receptor. Its action may contribute to the understanding of pain pathways and immune response modulation.

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Specifications

Manufacturer	Adooq Bioscience
Actions	Antagonist
CAS Number	3116848-78-0
Applications	MrgprX2 Antagonist
Formula	C₂₆H₂₆F₂N₈O₃
Molecular Weight	536.53
SMILES	O=C(N1C(C)(CN(CC1)[C@@H](C)C(NC2=NC=C(OC3=C(C=C(C=C3)F)F)N=C2)=O)C)C4=CC5=NC=NN5C=C4

Storage & Solubility

In Vitro Solubility

Reported Solubility

No reported solubility data are available for this product.

Preparing Stock Solutions

Stock preparation is unavailable for this product molecular weight.

Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.

Storage

Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.