Fig. 1 · Structure
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MRP1-IN-1
MRP1 Inhibitor
MRP1-IN-1 is a potent MRP1 inhibitor, exhibiting an EC50 of 0.90 μM in HeLa-T5 cells. This compound is instrumental in studying the modulation of multidrug resistance protein 1 (MRP1) and can be utilized in research related to drug transport mechanisms and cancer therapies. Its ability to inhibit MRP1 provides valuable insights into strategies for overcoming drug resistance in various malignancies.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Inhibitor |
| CAS Number | 246238-55-1 |
| Applications | MRP1 Inhibitor |
| Formula | C28H24ClN3O6 |
| Molecular Weight | 533.96 |
| SMILES | O=C1C2=C(C)ON=C2C3=C(N1C4=CC=CC(CC(NC5=CC(OC)=C(C(OC)=C5)OC)=O)=C4)C=CC=C3Cl |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.