MSC2530818

Catalog No.: A12644

CDK8 inhibitor

MSC2530818

MSC2530818 Chemical Structure

CAS NO. 1883423-59-3

MSC2530818 is a potent, selective and orally available CDK8 inhibitor with an IC50 of 2.6 nM for CDK8.

Availability: In stock

Package Price Qty
5 mg
$144.00
10 mg
$248.00
50 mg
$736.00
100 mg
$1,472.00
Custom Size Get quote

Free Overnight Delivery on orders over $500

Next day delivery by 10:00 a.m. Order now.

Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

MSC2530818 is a potent, selective and orally available CDK8 inhibitor with an IC50 of 2.6 nM for CDK8.
In vitro DMSO 66 mg/mL (193.65 mM)
Water Insoluble
Ethanol 66 mg/mL (193.65 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 29.34 mL 146.71 mL 293.42 mL
0.5 mM 5.87 mL 29.34 mL 58.68 mL
1 mM 2.93 mL 14.67 mL 29.34 mL
5 mM 0.59 mL 2.93 mL 5.87 mL

*The above data is based on the productmolecular weight 340.81. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A12644
Actions Inhibitor
CAS No. 1883423-59-3
Formula C18H17ClN4O
M. Wt 340.81
Solubility DMSO
Purity >98%
Synonyms MSC-2530818; MSC 2530818
SMILES O=C(N1[[email protected]](C2=CC=C(Cl)C=C2)CCC1)C3=CN=C(NN=C4C)C4=C3
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

Product Tags

Product Tags

Use spaces to separate tags. Use single quotes (') for phrases.

Product Questions

Product Questions

No Questions
Keywords:buy MSC2530818 | MSC2530818 Supplier | purchase | cost | manufacturer | order | distributor | buy 1883423-59-3| 1883423-59-3 Supplier | purchase 1883423-59-3 | 1883423-59-3 cost | 1883423-59-3 manufacturer | order 1883423-59-3 | 1883423-59-3 distributor
Rewards