Catalog No.: A12644

CDK8 inhibitor


MSC2530818 Chemical Structure

CAS NO. 1883423-59-3

MSC2530818 is a potent, selective and orally available CDK8 inhibitor with an IC50 of 2.6 nM for CDK8.

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Biological Activity

MSC2530818 is a potent, selective and orally available CDK8 inhibitor with an IC50 of 2.6 nM for CDK8.
In vitro DMSO 66 mg/mL (193.65 mM)
Water Insoluble
Ethanol 66 mg/mL (193.65 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 29.34 mL 146.71 mL 293.42 mL
0.5 mM 5.87 mL 29.34 mL 58.68 mL
1 mM 2.93 mL 14.67 mL 29.34 mL
5 mM 0.59 mL 2.93 mL 5.87 mL

*The above data is based on the productmolecular weight 340.81. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A12644
Actions Inhibitor
CAS No. 1883423-59-3
Formula C18H17ClN4O
M. Wt 340.81
Purity >98%
Synonyms MSC-2530818; MSC 2530818
SMILES O=C(N1[[email protected]](C2=CC=C(Cl)C=C2)CCC1)C3=CN=C(NN=C4C)C4=C3

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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