Fig. 1 · Structure
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N-Desalkylflurazepam
Benzodiazepine Metabolite
N-Desalkylflurazepam, a long-acting metabolite of benzodiazepine compounds like Flurazepam, primarily targets L-type voltage-gated calcium channels. It demonstrates inhibitory activity with IC50 values of 55 μM for Cav1.2 and 37 μM for Cav1.3. This compound is relevant in studies exploring nervous system modulation and the pharmacological effects of benzodiazepine metabolites in psychopharmacology and anxiety research.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| CAS Number | 2886-65-9 |
| Applications | Benzodiazepine Metabolite |
| Formula | C15H10ClFN2O |
| Molecular Weight | 288.70 |
| Synonyms | Norfludiazepam |
| SMILES | O=C1NC2=C(C(C3=C(F)C=CC=C3)=NC1)C=C(Cl)C=C2 |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.