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Biological Activity
Naftopidil 2HCl is a selective 5-HT1A and α1-adrenergic receptor antagonist with IC50 of 0.1 μM and 0.2 μM, respectively.
Targets
| 5-HT1A | α1-adrenergic receptor | |||
| 0.1 μM | 0.2 μM |
| In vitro (25°C) | DMSO | 35 mg/mL (75.2 mM) | |
| Water | Insoluble | ||
| Ethanol | 2 mg/mL (4.29 mM) | ||
| In vivo | 0.5% CMC | 28 mg/mL | |
|
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
|||
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 0.1 mM | 21.49 mL | 107.43 mL | 214.87 mL |
| 0.5 mM | 4.3 mL | 21.49 mL | 42.97 mL |
| 1 mM | 2.15 mL | 10.74 mL | 21.49 mL |
| 5 mM | 0.43 mL | 2.15 mL | 4.3 mL |
*The above data is based on the productmolecular weight 465.4 . Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
| Catalog Num | A10619 |
|---|---|
| Actions | Antagonist |
| CAS No. | 57149-08-3 |
| Formula | C24H28N2O3.2HCl |
| M. Wt | 465.4 |
| Purity | >98% |
| Synonyms | Flivas, KT-611, Avishot |
| SMILES | COC1=CC=CC=C1N2CCN(CC2)CC(COC3=CC=CC4=CC=CC=C43)O.Cl.Cl |
| Storage | Store lyophilized at -20ºC, keep desiccated. |
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