NaV1.2/1.6 channel blocker-1

Catalog No.: A68471
NaV1.2/1.6 Channel Blocker
NaV1.2/1.6 channel blocker-1 is a selective inhibitor of the NaV1.2 and NaV1.6 sodium channels, exhibiting IC50 values of 9.8 μM for rNaV1.6 and 24.4 μM for hNaV1.2. This compound is valuable for studying the role of sodium channels in neuronal excitability and has potential applications in the research of generalized epilepsy.
Grouped product items
Size Price Stock Qty
1mg
$25.00
In stock
5mg
$65.00
In stock
10mg
$100.00
In stock
25mg
$200.00
In stock
50mg
$290.00
In stock
100mg
$420.00
In stock
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Free Delivery on orders over $500
Research use only. We do not sell to patients.

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Adooq Products cited in reputable paper
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Nature Volume 622 Issue 7982 (2023)
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Biological Activity
DescriptionNaV1.2/1.6 channel blocker-1 is a selective inhibitor of the NaV1.2 and NaV1.6 sodium channels, exhibiting IC50 values of 9.8 μM for rNaV1.6 and 24.4 μM for hNaV1.2. This compound is valuable for studying the role of sodium channels in neuronal excitability and has potential applications in the research of generalized epilepsy.
Product Information
Catalog NumA68471
FormulaC14H14N2OS
Molecular Weight258.34
CAS Number1199944-04-1
SMILESS=C1OC2=CC=CC=C2C3=NC(C)=C(CCC)N13
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