Fig. 1 · Structure
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NCGC00135472
DRV1 Agonist
NCGC00135472 is a potent agonist of the resolvin D1 receptor (DRV1), exhibiting an EC50 of 0.37 nM for β-arrestin recruitment and 0.05 μM for cAMP activity. This compound plays a significant role in mediating anti-inflammatory responses and promoting resolution of inflammation. Its pharmacological properties make it a valuable tool for research applications focused on inflammation and resolution pathways in various biological contexts.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Agonist |
| CAS Number | 862811-76-5 |
| Applications | DRV1 Agonist |
| Formula | C20H14F2N4O |
| Molecular Weight | 364.35 |
| SMILES | O=C(NC1=CC=CC(C2=C(C)N3C=CC=NC3=N2)=C1)C4=CC=C(F)C(F)=C4 |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.