Nelotanserin

Catalog No.: A21506

5-HT2A inverse agonist

Nelotanserin

Nelotanserin Chemical Structure

CAS NO. 839713-36-9

Nelotanserin is a potent 5-HT2A inverse agonist, a moderately potent 5-HT2C partial inverse agonist and a weak 5-HT2B inverse agonist, with IC50s of 1.7, 79, 791 nM in IP accumulation assays, respectively.

Availability: In stock

Package Price Qty
5 mg
$90.00
10 mg
$155.00
50 mg
$460.00
100 mg
$920.00
Custom Size Get quote

Free Overnight Delivery on orders over $500

Next day delivery by 10:00 a.m. Order now.

Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

Nelotanserin is a potent 5-HT2A inverse agonist, a moderately potent 5-HT2C partial inverse agonist and a weak 5-HT2B inverse agonist, with IC50s of 1.7, 79, 791 nM in IP accumulation assays, respectively.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 22.87 mL 114.35 mL 228.71 mL
0.5 mM 4.57 mL 22.87 mL 45.74 mL
1 mM 2.29 mL 11.44 mL 22.87 mL
5 mM 0.46 mL 2.29 mL 4.57 mL

*The above data is based on the productmolecular weight 437.24. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A21506
Actions Agonist
M. Wt 437.24
Formula C18H15BrF2N4O2
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 839713-36-9
Synonyms APD125, APD 125, APD-125
SMILES COC1=C(C2=C(Br)C=NN2C)C=C(NC(NC3=C(F)C=C(F)C=C3)=O)C=C1

Product Tags

Product Tags

Use spaces to separate tags. Use single quotes (') for phrases.

Product Questions

Product Questions

No Questions
Keywords:buy Nelotanserin | Nelotanserin Supplier | purchase | cost | manufacturer | order | distributor | buy 839713-36-9| 839713-36-9 Supplier | purchase 839713-36-9 | 839713-36-9 cost | 839713-36-9 manufacturer | order 839713-36-9 | 839713-36-9 distributor
Rewards