Nepicastat (free base) (SYN-117)

Catalog No.: A10637

dopamine beta-hydroxylase inhibitor

Nepicastat (free base) (SYN-117)

Nepicastat (free base) (SYN-117) Chemical Structure

CAS NO. 173997-05-2

Nepicastat is an inhibitor of dopamine beta-hydroxylase, an enzyme that catalyzes the conversion of dopamine to norepinephrine.

Availability: In stock

Package Price Qty
5 mg
$150.00
10 mg
$270.00
50 mg
$718.00
100 mg
$1,300.00
Custom Size Get quote

Free Overnight Delivery on orders over $500

Next day delivery by 10:00 a.m. Order now.

Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

Nepicastat is an inhibitor of dopamine beta-hydroxylase, an enzyme that catalyzes the conversion of dopamine to norepinephrine.
In vitro (25°C) DMSO 61 mg/mL (183.83 mM)
Water Insoluble
Ethanol Insoluble
In vivo 30% propylene glycol, 5% Tween 80, 65% D5W 28 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 33.85 mL 169.26 mL 338.52 mL
0.5 mM 6.77 mL 33.85 mL 67.7 mL
1 mM 3.39 mL 16.93 mL 33.85 mL
5 mM 0.68 mL 3.39 mL 6.77 mL

*The above data is based on the productmolecular weight 295.4 . Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A10637
Actions Inhibitor
CAS No. 173997-05-2
Formula C14H15F2N3S
M. Wt 295.4
Solubility DMSO
Purity >98%
Synonyms RS-25560-197, SYN117
SMILES C1CC2=C(C=C(C=C2C[[email protected]]1N3C(=CNC3=S)CN)F)F
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

Product Tags

Product Tags

Use spaces to separate tags. Use single quotes (') for phrases.

Product Questions

Product Questions

No Questions
Keywords:buy Nepicastat (free base) (SYN-117) | Nepicastat (free base) (SYN-117) Supplier | purchase | cost | manufacturer | order | distributor | buy 173997-05-2| 173997-05-2 Supplier | purchase 173997-05-2 | 173997-05-2 cost | 173997-05-2 manufacturer | order 173997-05-2 | 173997-05-2 distributor
Rewards