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NR4A1 agonist 1

NR4A1 Agonist

NR4A1 Agonist 1 is a selective agonist of the NR4A1 receptor, exhibiting a Ki value of 2.96 μM. It demonstrates significant lipid-lowering effects in 3T3-L1 adipocytes, with an EC50 of 0.13 μM, leading to reduced triglyceride and lipid droplet accumulation. This compound is valuable for research applications focused on obesity and metabolic disorders.

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Specifications

Manufacturer	Adooq Bioscience
Actions	Agonist
CAS Number	1825366-87-7
Applications	NR4A1 Agonist
Formula	C₂₂H₂₃N₅O
Molecular Weight	373.45
SMILES	CN(CCCNC1=NC(C2=C(C3=CC=CC=C3N2)C=O)=NC4=C1C=CC=C4)C

Storage & Solubility

In Vitro Solubility

Reported Solubility

No reported solubility data are available for this product.

Preparing Stock Solutions

Stock preparation is unavailable for this product molecular weight.

Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.

Storage

Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.