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NSD2-IN-4

NSD2-SET inhibitor

NSD2-IN-4 is a selective inhibitor of the NSD2-SET domain, demonstrating strong efficacy in modulating histone methylation. This compound is particularly relevant in the study of NSD2-related diseases, including certain types of cancer, by targeting the dysregulation of epigenetic markers. Its utility in research underscores its potential for elucidating the biological mechanisms associated with NSD2 activity.

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Specifications

Manufacturer	Adooq Bioscience
Actions	Inhibitor
CAS Number	3035028-80-6
Applications	NSD2-SET inhibitor
Formula	C₁₈H₁₄ClN₃O₃
Molecular Weight	355.78
SMILES	O=C1C(NC2(C3)CC3(NC(C#CC)=O)C2)=C(Cl)C(C4=NC=CC=C41)=O

Storage & Solubility

In Vitro Solubility

Reported Solubility

No reported solubility data are available for this product.

Preparing Stock Solutions

Stock preparation is unavailable for this product molecular weight.

Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.

Storage

Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.