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Octoclothepine

Neuroleptic/Antipsychotic

Octoclothepine is a neuroleptic and antipsychotic agent that functions through dual enantiomeric forms—(+)-Octoclothepine and (-)-Octoclothepine. The (+)-form demonstrates exceptionally high binding affinity to 5-HT₆ and 5-HT₇ receptors, with Ki values of 0.41 nM and 0.38 nM, respectively, while the (-)-form shows Ki values of 17.7 nM and 1.3 nM. This compound is valuable in research focused on schizophrenia, exploring its atypical and typical antipsychotic properties.

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Specifications

Manufacturer	Adooq Bioscience
CAS Number	13448-22-1
Applications	Neuroleptic/Antipsychotic
Formula	C₁₉H₂₁ClN₂S
Molecular Weight	344.90
Synonyms	Clorotepine
SMILES	CN1CCN(C2CC3=CC=CC=C3SC4=CC=C(Cl)C=C24)CC1

Storage & Solubility

In Vitro Solubility

Reported Solubility

No reported solubility data are available for this product.

Preparing Stock Solutions

Stock preparation is unavailable for this product molecular weight.

Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.

Storage

Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.