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Biological Activity
Oxprenolol is an orally bioavailable β-adrenergic receptor (β-AR) antagonist (Ki = 7.10 nM in a radioligand binding assay using rat heart tissue). It is non-selective and inhibits both β1- and β2-ARs (Kds = 2.09 and 1.35 nM in isolated rat heart and uterus, respectively). Oxprenolol is selective for β-ARs over serotonin (5-HT) receptors in rat sarcolemmal membrane preparations (IC50s = 4.13 and 23,300 nM, respectively), but it binds to 5-HT1A receptors in rat hippocampus and 5-HT1B in rat striatum (Kis = 94.2 and 642 nM, respectively).
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 0.1 mM | 33.13 mL | 165.67 mL | 331.33 mL |
| 0.5 mM | 6.63 mL | 33.13 mL | 66.27 mL |
| 1 mM | 3.31 mL | 16.57 mL | 33.13 mL |
| 5 mM | 0.66 mL | 3.31 mL | 6.63 mL |
*The above data is based on the productmolecular weight 301.81. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
| Catalog Num | A17368 |
|---|---|
| Actions | Antagonist |
| CAS No. | 6452-73-9 |
| Formula | C15H24ClNO3 |
| M. Wt | 301.81 |
| Purity | >98% |
| Synonyms | Oxprenolol hydrochloride; Coretal; Dialicor; Rixiprol; Trasicor; Evinrozit; Ranidrox; Oxprenolol HCl; Trepress; Vrachor; Ba 39089; Ba-39089; Ba39089 |
| SMILES | OC(CNC(C)C)COC1=CC=CC=C1OCC=C.[H]Cl |
| Storage | Store lyophilized at -20ºC, keep desiccated. |
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