Biological Activity
PD-159020 is a non-selective ETA/ETB antagonist, with IC50s of 30 and 50 nM for hETA and hETB, respectively.
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
---|---|---|---|
0.1 mM | 18.13 mL | 90.66 mL | 181.31 mL |
0.5 mM | 3.63 mL | 18.13 mL | 36.26 mL |
1 mM | 1.81 mL | 9.07 mL | 18.13 mL |
5 mM | 0.36 mL | 1.81 mL | 3.63 mL |
*The above data is based on the productmolecular weight 551.54. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
Catalog Num | A13499 |
---|---|
Actions | Antagonist |
CAS No. | 177904-00-6 |
Formula | C32H25NO8 |
M. Wt | 551.54 |
Solubility | DMSO |
Purity | >98% |
Synonyms | PD159020, PD159020 |
SMILES | O=C(C(N1CC2=CC=C(OCO3)C3=C2)=C(C4=CC=C(OCO5)C5=C4)C6=C1C=C(OCC7=CC=CC=C7)C(OC)=C6)O |
Storage | Store lyophilized at -20ºC, keep desiccated. |
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