Fig. 1 · Structure
Documents & Downloads
PDK1 allosteric modulator 1
PDK-1 Modulator
PDK1 Allosteric Modulator 1 is a selective compound targeting the PDK1 kinase through allosteric modulation, exhibiting a binding affinity of 8 μM. By interacting with the PIF pocket of PDK1, this modulator can influence the enzyme's biological activity. It is suitable for research applications focused on understanding PDK1's role in cellular signaling pathways and the development of therapeutics targeting related conditions.
In Stock
Free Aliquoting for Your Order
Tell us your preferred amount per vial. We’ll confirm the options.
Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Modulator |
| CAS Number | 303134-93-2 |
| Applications | PDK-1 Modulator |
| Formula | C17H15FN2O3S |
| Molecular Weight | 346.38 |
| SMILES | O=C(CN1C(SCCOC2=C(F)C=CC=C2)=NC3=C1C=CC=C3)O |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.