PF-03382792 is a potent partial agonist of the 5-HT4 receptor, exhibiting a Ki value of 2.7 nM and an EC50 of 0.9 nM for the 5-HT4d subtype. This compound demonstrates the ability to penetrate the blood-brain barrier and has been shown to elicit moderate increases in cortical acetylcholine levels in the rat prefrontal cortex. PF-03382792 is a valuable tool for research investigating cognitive processes and potential therapeutic strategies for neurological disorders.
PF-03382792 is a potent partial agonist of the 5-HT4 receptor, exhibiting a Ki value of 2.7 nM and an EC50 of 0.9 nM for the 5-HT4d subtype. This compound demonstrates the ability to penetrate the blood-brain barrier and has been shown to elicit moderate increases in cortical acetylcholine levels in the rat prefrontal cortex. PF-03382792 is a valuable tool for research investigating cognitive processes and potential therapeutic strategies for neurological disorders.
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