PF-07258669 is a potent orally active antagonist of the melanocortin-4 receptor (MC4R), displaying an IC50 of 13 nM and a Ki of 0.46 nM. This compound has significant implications for research into conditions related to cachexia, anorexia, and anorexia nervosa, making it a valuable tool for studying the regulatory mechanisms of appetite and energy homeostasis.
PF-07258669 is a potent orally active antagonist of the melanocortin-4 receptor (MC4R), displaying an IC50 of 13 nM and a Ki of 0.46 nM. This compound has significant implications for research into conditions related to cachexia, anorexia, and anorexia nervosa, making it a valuable tool for studying the regulatory mechanisms of appetite and energy homeostasis.
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