PF-4522654 is a selective agonist of the 5-HT2C receptor, exhibiting a potent EC50 of 16 nM and a Ki of 8 nM. This compound demonstrates negligible functional activity at the 5-HT2A and 5-HT2B receptors, thereby ensuring specificity. PF-4522654 is employed in research focused on stress urinary incontinence (SUI), making it a valuable tool for exploring potential therapeutic approaches in this area.
PF-4522654 is a selective agonist of the 5-HT2C receptor, exhibiting a potent EC50 of 16 nM and a Ki of 8 nM. This compound demonstrates negligible functional activity at the 5-HT2A and 5-HT2B receptors, thereby ensuring specificity. PF-4522654 is employed in research focused on stress urinary incontinence (SUI), making it a valuable tool for exploring potential therapeutic approaches in this area.
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