PF-915275

Catalog No.: A21330

11βHSD1 inhibitor

PF-915275

PF-915275 Chemical Structure

CAS NO. 857290-04-1

PF-915275 is a potent, selective and orally active human 11β-hydroxysteroid dehydrogenase type 1 (11βHSD1) inhibitor with a Ki of 2.3 nM and an EC50 of 15 nM (in HEK293 cells).

Availability: In stock

Package Price Qty
5 mg
$97.00
10 mg
$167.00
50 mg
$497.00
100 mg
$994.00
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Biological Activity

PF-915275 is a potent, selective and orally active human 11β-hydroxysteroid dehydrogenase type 1 (11βHSD1) inhibitor with a Ki of 2.3 nM and an EC50 of 15 nM (in HEK293 cells).
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 28.54 mL 142.7 mL 285.4 mL
0.5 mM 5.71 mL 28.54 mL 57.08 mL
1 mM 2.85 mL 14.27 mL 28.54 mL
5 mM 0.57 mL 2.85 mL 5.71 mL

*The above data is based on the productmolecular weight 350.39. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A21330
Actions Inhibitor
M. Wt 350.39
Formula C18H14N4O2S
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 857290-04-1
SMILES N#CC1=CC=C(C2=CC=C(S(NC3=NC(N)=CC=C3)(=O)=O)C=C2)C=C1

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