Fig. 1 · Structure
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PI5P4Kγ-IN-1
PI5P4Kγ Inhibitor
PI5P4Kγ-IN-1 is a highly selective inhibitor that targets PI5P4Kγ through an ATP-competitive mechanism, exhibiting a Kd of 19 nM and an IC50 of 67 nM. This compound effectively inhibits the function of PI5P4Kγ and enhances the mTORC1 signaling pathway in cellular contexts. PI5P4Kγ-IN-1 is valuable for research applications in understanding the role of PI5P4Kγ in various diseases, including breast cancer.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Inhibitor |
| CAS Number | 2419358-87-3 |
| Applications | PI5P4Kγ Inhibitor |
| Formula | C20H20N4O |
| Molecular Weight | 332.40 |
| SMILES | NC1=NC(C2=C(CCC3)NC4=C2C=C(C5=CCOCC5)C=C4)=C3C=N1 |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.