Pimozide

Catalog No.: A17375

Dopamine receptor antagonist

Pimozide

Pimozide Chemical Structure

CAS NO. 2062-78-4

Pimozide is a dopamine receptor antagonist, with Kis of 1.4 nM, 2.5 nM and 588 nM for dopamine D2, D3 and D1 receptors, respectively, and also has affinity at α1-adrenoceptor, with a Ki of 39 nM; Pimozide also inhibits STAT3 and STAT5.

Availability: In stock

Package Price Qty
50 mg
$45.00
100 mg
$80.00
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Warning WARNING: Attention California Residents: This product can expose you to chemicals including Pimozide , which is known to the State of California to cause cancer and birth defects or other reproductive harm. For more information, go to www.P65Warnings.ca.gov
Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

Pimozide is a dopamine receptor antagonist, with Kis of 1.4 nM, 2.5 nM and 588 nM for dopamine D2, D3 and D1 receptors, respectively, and also has affinity at α1-adrenoceptor, with a Ki of 39 nM; Pimozide also inhibits STAT3 and STAT5.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 21.67 mL 108.33 mL 216.66 mL
0.5 mM 4.33 mL 21.67 mL 43.33 mL
1 mM 2.17 mL 10.83 mL 21.67 mL
5 mM 0.43 mL 2.17 mL 4.33 mL

*The above data is based on the productmolecular weight 461.55. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A17375
Actions Antagonist
M. Wt 461.55
Formula C28H29F2N3O
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 2062-78-4
Synonyms R 6238; R-6238; R6238; Pimozide; Orap; Opiran.
SMILES O=C1N(C2CCN(CCCC(C3=CC=C(F)C=C3)C4=CC=C(F)C=C4)CC2)C5=CC=CC=C5N1

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