Documents & Downloads

Pitolisant-d6

Stable Isotope

Pitolisant-d6 is a deuterium-labeled derivative of Pitolisant, which acts as a potent and selective nonimidazole inverse agonist at the recombinant human histamine H3 receptor (Ki=0.16 nM). This stable isotope-labeled compound is utilized in pharmacokinetic studies and metabolic research, allowing for in-depth analysis of drug metabolism and interaction with the H3 receptor. It is an essential tool for researchers investigating sleep disorders and cognitive function modulation.

Out of Stock

Free Aliquoting for Your Order

Tell us your preferred amount per vial. We’ll confirm the options.

Specifications

Manufacturer	Adooq Bioscience
CAS Number	2416991-77-8
Applications	Stable Isotope
Formula	C₁₇H₂₀D₆ClNO
Molecular Weight	301.88
Synonyms	Tiprolisant-d6
SMILES	[2H]C(N1CCCCC1)([2H])C([2H])([2H])C([2H])([2H])OCCCC2=CC=C(C=C2)Cl

Storage & Solubility

In Vitro Solubility

Reported Solubility

No reported solubility data are available for this product.

Preparing Stock Solutions

Stock preparation is unavailable for this product molecular weight.

Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.

Storage

Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.