Prazobind-d8 is a deuterium-labeled analog of Prazobind, functioning as an irreversible antagonist of the α1-adrenoceptor. With an IC50 value of 1 nM, Prazobind-d8 exhibits potent competitive binding to α1-adrenoceptor subtypes, specifically in the hippocampus and liver. This compound partially inhibits contractions in smooth, circular, and longitudinal muscle tissues, making it a valuable tool for investigating mechanisms related to blood pressure regulation and related cardiovascular research.
Prazobind-d8 is a deuterium-labeled analog of Prazobind, functioning as an irreversible antagonist of the α1-adrenoceptor. With an IC50 value of 1 nM, Prazobind-d8 exhibits potent competitive binding to α1-adrenoceptor subtypes, specifically in the hippocampus and liver. This compound partially inhibits contractions in smooth, circular, and longitudinal muscle tissues, making it a valuable tool for investigating mechanisms related to blood pressure regulation and related cardiovascular research.
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