PROTAC ERRα ligand 2

Catalog No.: A18939

ERRα inverse agonist

PROTAC ERRα ligand 2

PROTAC ERRα ligand 2 Chemical Structure

CAS NO. 2306388-57-6

PROTAC ERRα ligand 2 is an estrogen-related receptor α (ERRα) inverse agonist with an IC50 of 5.67 nM. PROTAC ERRα ligand 2 (IC50=5.67 nM) displays a ~11-fold improved potency than XCT790 (IC50=61.3 nM).

Availability: In stock

Package Price Qty
5 mg

Regular Price: $270.00

Special Price $216.00

10 mg

Regular Price: $465.00

Special Price $372.00

50 mg

Regular Price: $1,380.00

Special Price $1,104.00

100 mg

Regular Price: $2,760.00

Special Price $2,208.00

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Biological Activity

PROTAC ERRα ligand 2 is an estrogen-related receptor α (ERRα) inverse agonist with an IC50 of 5.67 nM. PROTAC ERRα ligand 2 (IC50=5.67 nM) displays a ~11-fold improved potency than XCT790 (IC50=61.3 nM).
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 22.46 mL 112.28 mL 224.56 mL
0.5 mM 4.49 mL 22.46 mL 44.91 mL
1 mM 2.25 mL 11.23 mL 22.46 mL
5 mM 0.45 mL 2.25 mL 4.49 mL

*The above data is based on the productmolecular weight 445.31. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A18939
Actions Agonist
CAS No. 2306388-57-6
Formula C20H13F6NO4
M. Wt 445.31
Purity >98%
Synonyms 0
SMILES O=C(O)/C(C#N)=C/C1=CC(OC)=C(C=C1)OCC2=CC=C(C(F)(F)F)C=C2C(F)(F)F
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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