Fig. 1 · Structure
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PSNCBAM-1
Cannabinoid Receptor Antagonist
PSNCBAM-1 is a selective allosteric antagonist of the cannabinoid receptor type 1 (CB1), with an EC50 of 0.1 μM. This compound serves as a valuable tool in the investigation of obesity and related metabolic disorders, providing insights into the modulation of cannabinoid signaling pathways. Its specificity for the CB1 receptor makes it suitable for exploring therapeutic approaches targeting endocannabinoid system regulation.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Antagonist |
| CAS Number | 877202-74-9 |
| Applications | Cannabinoid Receptor Antagonist |
| Formula | C22H21ClN4O |
| Molecular Weight | 392.88 |
| SMILES | ClC(C=C1)=CC=C1NC(NC2=CC=CC(C3=CC=CC(N4CCCC4)=N3)=C2)=O |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.