Customer Appreciation Sale.
15% off with promo code "APPRECIATION2023" on check out or purchase order

Pyrotinib dimaleate

Catalog No.: A21756

EGFR/HER2 dual inhibitor

Pyrotinib dimaleate

Pyrotinib dimaleate Chemical Structure

CAS NO. 1397922-61-0

Pyrotinib dimaleate (SHR-1258 dimaleate) is a potent and selective EGFR/HER2 dual inhibitor with IC50 s of 13 and 38 nM, respectively.

Availability: In stock

Package Price Qty
1 mg
$205.00
5 mg
$616.00
10 mg
$1,049.00
50 mg
$3,146.00
Custom Size Get quote

Free Overnight Delivery on orders over $500

Next day delivery by 10:00 a.m. Order now.

Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

Pyrotinib dimaleate (SHR-1258 dimaleate) is a potent and selective EGFR/HER2 dual inhibitor with IC50 s of 13 and 38 nM, respectively.
In vitro DMSO Insoluble
Water Insoluble
Ethanol Insoluble
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 12.27 mL 61.33 mL 122.67 mL
0.5 mM 2.45 mL 12.27 mL 24.53 mL
1 mM 1.23 mL 6.13 mL 12.27 mL
5 mM 0.25 mL 1.23 mL 2.45 mL

*The above data is based on the productmolecular weight 815.22. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A21756
Actions Inhibitor
CAS No. 1397922-61-0
Formula C40H39ClN6O11
M. Wt 815.22
Purity >98%
Synonyms SHR-1258 dimaleate, SHR1258, SHR 1258
SMILES O=C(NC1=C(OCC)C=C2N=CC(C#N)=C(NC3=CC=C(OCC4=NC=CC=C4)C(Cl)=C3)C2=C1)/C=C/[[email protected]@H]5N(C)CCC5.O=C(O)/C=C\C(O)=O.O=C(O)/C=C\C(O)=O
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

Product Tags

Product Tags

Use spaces to separate tags. Use single quotes (') for phrases.

Product Questions

Product Questions

No Questions
Keywords:buy Pyrotinib dimaleate | Pyrotinib dimaleate Supplier | purchase | cost | manufacturer | order | distributor | buy 1397922-61-0| 1397922-61-0 Supplier | purchase 1397922-61-0 | 1397922-61-0 cost | 1397922-61-0 manufacturer | order 1397922-61-0 | 1397922-61-0 distributor
Rewards