Fig. 1 · Structure
Documents & Downloads
Quipazine dimaleate
5-HT Agonist
Quipazine dimaleate is a potent 5-HT agonist, demonstrating a Ki value of 1.4 nM for displacing [3H]GR65630 from the 5-HT3 receptor in rat models. This compound exhibits antiviral activity against SARS-CoV-2, with an EC50 of 31.64 μM, and acts as a 5-HT3 receptor antagonist in peripheral models. Quipazine dimaleate is valuable for research in neurological diseases, providing insights into serotonin receptor modulation and antiviral mechanisms.
In Stock
Free Aliquoting for Your Order
Tell us your preferred amount per vial. We’ll confirm the options.
Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Agonist |
| CAS Number | 150323-78-7 |
| Applications | 5-HT Agonist |
| Formula | C21H23N3O8 |
| Molecular Weight | 445.42 |
| SMILES | O=C(O)/C=C\C(O)=O.O=C(O)/C=C\C(O)=O.C1(N2CCNCC2)=NC3=CC=CC=C3C=C1 |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.