Fig. 1 · Structure
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(Rac)-CPI-203
CPI-203 Racemate
(Rac)-CPI-203 is a racemic mixture of the bromodomain inhibitor CPI-203, which targets the BET (bromodomain and extraterminal domain) family of proteins. This compound exhibits significant biological activity by inhibiting the interaction between BET proteins and acetylated histones, thereby affecting gene expression regulation. It is utilized in research applications focused on cancer biology, inflammation, and epigenetic regulation, making it a valuable tool for studying signal transduction pathways and therapeutic intervention in various diseases.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Inhibitor |
| CAS Number | 202591-23-9 |
| Applications | CPI-203 Racemate |
| Formula | C19H18ClN5OS |
| Molecular Weight | 399.90 |
| SMILES | ClC1=CC=C(C2=NC(CC(N)=O)C3=NN=C(C)N3C4=C2C(C)=C(C)S4)C=C1 |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.