Documents & Downloads

(Rac)-GSK2973980A

DGAT1 Inhibitor

(Rac)-GSK2973980A is a potent diacylglycerol acyltransferase 1 (DGAT1) inhibitor with an IC50 of 1.8 nM for human DGAT1. This compound is useful for investigating the role of DGAT1 in lipid metabolism and is applicable in obesity and obesity-related disease research. Its selective inhibition of DGAT1 provides valuable insights into therapeutic targets for metabolic disorders.

Out of Stock

Free Aliquoting for Your Order

Tell us your preferred amount per vial. We’ll confirm the options.

Specifications

Manufacturer	Adooq Bioscience
Actions	Inhibitor
CAS Number	1414797-35-5
Applications	DGAT1 Inhibitor
Formula	C₂₅H₁₉F₅N₄O₄
Molecular Weight	534.44
SMILES	O=C(O)CC1(C(=O)C2=CC=C(C=C2CC1)C3=NC=C(N=C3)NC(=O)NC4=CC=C(F)C(F)=C4)CC(F)(F)F

Storage & Solubility

In Vitro Solubility

Reported Solubility

No reported solubility data are available for this product.

Preparing Stock Solutions

Stock preparation is unavailable for this product molecular weight.

Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.

Storage

Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.