Fig. 1 · Structure
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RBI-257 maleate
Dopamine D4 Receptor Antagonist
RBI-257 maleate is a potent antagonist of the dopamine D4 receptor, exhibiting a Ki value of 0.3 nM. This compound has demonstrated significant biological activity in modulating dopaminergic signaling and is valuable for research applications related to neuropharmacology and psychiatric disorders. Its selectivity for the D4 receptor makes it a suitable tool for investigating the role of dopamine in various behavioral and neurological models.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Antagonist |
| CAS Number | 911378-38-6 |
| Applications | Dopamine D4 Receptor Antagonist |
| Formula | C25H32IN3O5 |
| Molecular Weight | 581.44 |
| SMILES | CC(C)OC1=CC=CN=C1N(C2CCN(CC3=CC=C(I)C=C3)CC2)C.O=C(O)/C=C\C(O)=O |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.