Fig. 1 · Structure
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Rec 15/2615 hydrochloride
α-1B Adrenoceptor Antagonist
Rec 15/2615 hydrochloride is a highly selective antagonist of the α-1B adrenoceptor, exhibiting Ki values of 1.9 nM, 0.3 nM, and 2.6 nM for α1A, α1B, and α1D receptors, respectively. This compound effectively modulates vaginal smooth muscle contractility and augments genital engorgement, making it a valuable tool for studying the physiological roles of α-1B adrenergic signaling. Its specificity and potency aid in elucidating the mechanisms underlying reproductive and vascular functions in various research applications.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Antagonist |
| CAS Number | 173059-17-1 |
| Applications | α-1B Adrenoceptor Antagonist |
| Formula | C26H34ClN5O5 |
| Molecular Weight | 532.03 |
| SMILES | CC(C1=C(OCC(N2CCN(C3=NC(N)=C4C=C(OC)C(OC)=CC4=N3)CC2)=O)C(OC)=CC=C1)C.[H]Cl |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.