Fig. 1 · Structure
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rel-Ceperognastat
O-GlcNAcase Inhibitor
rel-Ceperognastat (rel-LY3372689) is a selective inhibitor of O-GlcNAcase (OGA), an important enzyme involved in the regulation of O-GlcNAcylation. By inhibiting OGA, rel-Ceperognastat enhances O-GlcNAc levels, thereby influencing various cellular processes. This compound is utilized in research focused on neurodegenerative diseases, including Alzheimer's disease, to explore its effects on neurobiology and potential therapeutic applications.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Inhibitor |
| CAS Number | 2241514-58-7 |
| Applications | O-GlcNAcase Inhibitor |
| Formula | C16H22FN5O3S |
| Molecular Weight | 383.44 |
| Synonyms | rel-LY3372689 |
| SMILES | CC(NC1=NC(F)=C(S1)CN2[C@@H](C[C@@H](CC2)OCC3=NOC(C)=N3)C)=O |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.