Fig. 1 · Structure
Documents & Downloads
Renzapride
5HT4 Receptor Agonist
Renzapride is a full agonist of the 5-HT4 receptor, exhibiting a Ki value of 115 nM. Additionally, it acts as an antagonist at both the 5-HT2b and 5-HT3 receptors. This compound is primarily utilized in research focusing on constipation-predominant irritable bowel syndrome (C-IBS), making it valuable for exploring therapeutic interventions in gastrointestinal disorders.
In Stock
Free Aliquoting for Your Order
Tell us your preferred amount per vial. We’ll confirm the options.
Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Agonist |
| CAS Number | 112727-80-7 |
| Applications | 5HT4 Receptor Agonist |
| Formula | C16H22ClN3O2 |
| Molecular Weight | 323.82 |
| Synonyms | BRL 24924 |
| SMILES | ClC1=C(N)C=C(OC)C(C(N[C@H]2CCN3CCC[C@@H]2C3)=O)=C1 |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.