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Rezatapopt analog-1

Rezatapopt Analog

Rezatapopt analog-1 is an analog of Rezatapopt, specifically targeting the TP53 Y220C mutation. This compound is designed to restore p53 tumor suppressor functions by stabilizing the protein's structure, thereby enhancing its biological activity against tumors with this specific mutation. Research applications include the study of p53-related pathways and therapeutic strategies for cancers harboring TP53 mutations.

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Specifications

Manufacturer	Adooq Bioscience
Actions	Inhibitor
CAS Number	2636846-37-0
Applications	Rezatapopt Analog
Formula	C₂₇H₂₈F₄N₄O₃
Molecular Weight	532.53
Synonyms	PC14586 analog-1
SMILES	FC(F)(F)CN1C2=CC=CC(N[C@H]3[C@H](CN(CC3)C)F)=C2C=C1C#CCNC4=C(C=C(C=C4)C(O)=O)OC

Storage & Solubility

In Vitro Solubility

Reported Solubility

No reported solubility data are available for this product.

Preparing Stock Solutions

Stock preparation is unavailable for this product molecular weight.

Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.

Storage

Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.