RGFP966

Catalog No.: A13218

HDAC3 inhibitor

RGFP966

RGFP966 Chemical Structure

CAS NO. 1357389-11-7

RGFP966 is an HDAC3 inhibitor with IC50 of 0.08 μM, exhibits > 200-fold selectivity over other HDAC.

Availability: In stock

Package Price Qty
5 mg
$90.00
10 mg
$140.00
25 mg
$270.00
50 mg
$350.00
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Biological Activity

RGFP966 is an HDAC3 inhibitor with IC50 of 0.08 μM, exhibits > 200-fold selectivity over other HDAC.
In vitro (25°C) DMSO 70 mg/mL (193.15 mM)
Water Insoluble
Ethanol Insoluble
In vivo 5%DMSO+40%PEG300+10%Tween80+45%ddH2O 6.1 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 27.59 mL 137.97 mL 275.94 mL
0.5 mM 5.52 mL 27.59 mL 55.19 mL
1 mM 2.76 mL 13.8 mL 27.59 mL
5 mM 0.55 mL 2.76 mL 5.52 mL

*The above data is based on the productmolecular weight 362.4. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A13218
Actions Inhibitor
CAS No. 1357389-11-7
Formula C21H19FN4O
M. Wt 362.4
Solubility DMSO
Purity >98%
Synonyms RGFP-966, RGFP 966
SMILES C1=CC=C(C=C1)/C=C/CN2C=C(C=N2)/C=C/C(=O)NC3=C(C=C(C=C3)F)N
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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