Rislenemdaz

Catalog No.: A21907

NMDA receptor GluN2B antagonist

Rislenemdaz

Rislenemdaz Chemical Structure

CAS NO. 808732-98-1

Rislenemdaz (CERC-301) is an orally bioavailable and selective N-methyl-D-aspartate (NMDA) receptor subunit 2B (GluN2B) antagonist with Ki and IC50 of 8.1 nM and 3.6 nM, respectively.

Availability: In stock

Package Price Qty
1 mg
$162.00
5 mg
$486.00
10 mg
$828.00
50 mg
$2,484.00
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Biological Activity

Rislenemdaz (CERC-301) is an orally bioavailable and selective N-methyl-D-aspartate (NMDA) receptor subunit 2B (GluN2B) antagonist with Ki and IC50 of 8.1 nM and 3.6 nM, respectively.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 27.9 mL 139.51 mL 279.01 mL
0.5 mM 5.58 mL 27.9 mL 55.8 mL
1 mM 2.79 mL 13.95 mL 27.9 mL
5 mM 0.56 mL 2.79 mL 5.58 mL

*The above data is based on the productmolecular weight 358.41. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A21907
Actions Antagonist
CAS No. 808732-98-1
Formula C19H23FN4O2
M. Wt 358.41
Solubility DMSO
Purity >98%
Synonyms MK-0657, MK0657, MK 0657; CERC-301, CERC 301, CERC301
SMILES O=C(N1C[[email protected]@H](F)[[email protected]@H](CNC2=NC=CC=N2)CC1)OCC3=CC=C(C)C=C3
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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