Roblitinib

Catalog No.: A19431

FGFR4 inhibitor

Roblitinib

Roblitinib Chemical Structure

CAS NO. 1708971-55-4

Roblitinib (FGF-401; Compound Example 83) is a highly selective and potent FGFR4 inhibitor with an IC50 of 1.9 nM. Roblitinib has antitumor activity.

Availability: In stock

Package Price Qty
2 mg
$80.00
5 mg
$120.00
10 mg
$200.00
50 mg
$600.00
Custom Size Get quote

Free Overnight Delivery on orders over $500

Next day delivery by 10:00 a.m. Order now.

Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

Roblitinib (FGF-401; Compound Example 83) is a highly selective and potent FGFR4 inhibitor with an IC50 of 1.9 nM. Roblitinib has antitumor activity.
In vitro DMSO 5 mg/mL (9.87 mM)
Water Insoluble
Ethanol 2 mg/mL (3.94 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 19.74 mL 98.7 mL 197.41 mL
0.5 mM 3.95 mL 19.74 mL 39.48 mL
1 mM 1.97 mL 9.87 mL 19.74 mL
5 mM 0.39 mL 1.97 mL 3.95 mL

*The above data is based on the productmolecular weight 506.56. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A19431
Actions Inhibitor
CAS No. 1708971-55-4
Formula C25H30N8O4
M. Wt 506.56
Purity >98%
Synonyms FGF-401, FGF401, FGF 401
SMILES CN1CC(N(CC2=CC(CCCN3C(NC4=CC(NCCOC)=C(C#N)C=N4)=O)=C3N=C2C=O)CC1)=O
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

Product Tags

Product Tags

Use spaces to separate tags. Use single quotes (') for phrases.

Product Questions

Product Questions

No Questions
Keywords:buy Roblitinib | Roblitinib Supplier | purchase | cost | manufacturer | order | distributor | buy 1708971-55-4| 1708971-55-4 Supplier | purchase 1708971-55-4 | 1708971-55-4 cost | 1708971-55-4 manufacturer | order 1708971-55-4 | 1708971-55-4 distributor
Rewards