RS-102221 is a selective antagonist of the 5-HT2C receptor, exhibiting a Ki value of 10 nM. This compound demonstrates significant selectivity, being nearly 100-fold more effective against the 5-HT2C receptor compared to the 5-HT2A and 5-HT2B receptors. RS-102221 has been shown to promote the differentiation of new nerve cells and is associated with increased food intake and weight gain in rat models, making it a valuable tool for research in neurobiology and metabolic studies.
RS-102221 is a selective antagonist of the 5-HT2C receptor, exhibiting a Ki value of 10 nM. This compound demonstrates significant selectivity, being nearly 100-fold more effective against the 5-HT2C receptor compared to the 5-HT2A and 5-HT2B receptors. RS-102221 has been shown to promote the differentiation of new nerve cells and is associated with increased food intake and weight gain in rat models, making it a valuable tool for research in neurobiology and metabolic studies.
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