Fig. 1 · Structure
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RS 39604
5-HT4 Receptor Antagonist
RS 39604 is a potent and selective antagonist of the 5-HT4 receptor, exhibiting a pKi of 9.1 in guinea pig striatal membranes. It demonstrates minimal affinity for other serotonin receptors, including 5-HT1A, 5-HT2C, and 5-HT3, as well as for various adrenergic, dopaminergic, muscarinic, angiotensin, and opioid receptors. RS 39604's distinctive profile makes it a valuable tool in research focusing on gastrointestinal motility disorders and neuropharmacology.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Antagonist |
| CAS Number | 167710-87-4 |
| Applications | 5-HT4 Receptor Antagonist |
| Formula | C26H37Cl2N3O6S |
| Molecular Weight | 590.56 |
| SMILES | CS(=O)(NCCN1CCC(CCC(C2=CC(Cl)=C(N)C=C2OCC3=CC(OC)=CC(OC)=C3)=O)CC1)=O.Cl |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.