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RSK4-IN-2

RSK4 Inhibitor

RSK4-IN-2 is a selective inhibitor of RSK4 with a potent inhibitory effect, demonstrating an IC50 of 17 nM. This compound effectively suppresses cell growth and invasion in esophageal squamous cell carcinoma (ESCC) by inhibiting the phosphorylation of RSK4 downstream targets. Additionally, RSK4-IN-2 has shown significant activity in reducing tumor growth and metastasis in ESCC mouse models, making it a valuable tool for research into ESCC development and progression.

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Specifications

Manufacturer	Adooq Bioscience
Actions	Inhibitor
CAS Number	3034203-03-4
Applications	RSK4 Inhibitor
Formula	C₁₇H₁₆N₈O
Molecular Weight	348.36
SMILES	O=C1N(C2=NC(NC3=CC=C4NN=NC4=C3)=NC=C2N=C1)C5CCCC5

Storage & Solubility

In Vitro Solubility

Reported Solubility

No reported solubility data are available for this product.

Preparing Stock Solutions

Stock preparation is unavailable for this product molecular weight.

Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.

Storage

Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.